CBP/p300-IN-2


Catalog No. Size PriceQuantity
M14001-2 Contact sales@xcessbio.com for quotation $100

Description

CBP/EP300-IN-2 is an inhibitor of CBP/EP300 with IC50 values of 1.07 nM and 5.96 nM for CBP/HTRF and Myc, respectively. CBP/EP300-IN-2, example 25, is extracted from patent WO2017205538A1.

Product information

CAS Number: 2158265-96-2

Molecular Weight: 521.56

Formula: C27H29F2N7O2

Chemical Name: 3-[6-(difluoromethyl)-7-(1-methyl-1H-pyrazol-4-yl)isoquinolin-4-yl]-N-methyl-1-(oxan-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide

Smiles: CN1C=C(C=N1)C1=CC2C=NC=C(C3=NN(C4CCOCC4)C4CCN(CC3=4)C(=O)NC)C=2C=C1C(F)F

InChiKey: ZDKBXFITPIXJAT-UHFFFAOYSA-N

InChi: InChI=1S/C27H29F2N7O2/c1-30-27(37)35-6-3-24-23(15-35)25(33-36(24)18-4-7-38-8-5-18)22-13-31-11-16-9-19(17-12-32-34(2)14-17)21(26(28)29)10-20(16)22/h9-14,18,26H,3-8,15H2,1-2H3,(H,30,37)

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

References:

  1. Patrick Cyr, et al. Pyrazolopyridine derivatives for the treatment of cancer

Products are for research use only. Not for human use.

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