GSK8573


Catalog No. Size PriceQuantity
M14336-2 2mg solid $150
M14336-10 10mg solid $460

Description

GSK8573 (compound 23) is an inactive control compound for GSK2801. GSK8573 has binding activity to BRD9 with a Kd value of 1.04 μM and is inactive against BAZ2A/B and other bromodomain familiy.

Product information

CAS Number: 1693766-04-9

Molecular Weight: 323.39

Formula: C20H21NO3

Chemical Name: 1-[1-(3-methoxyphenyl)-7-propoxyindolizin-3-yl]ethan-1-one

Smiles: CC(=O)C1=CC(=C2C=C(C=CN21)OCCC)C1C=C(C=CC=1)OC

InChiKey: QQBGNWWJANJWNY-UHFFFAOYSA-N

InChi: InChI=1S/C20H21NO3/c1-4-10-24-17-8-9-21-19(14(2)22)13-18(20(21)12-17)15-6-5-7-16(11-15)23-3/h5-9,11-13H,4,10H2,1-3H3

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Solubility: DMSO : 25 mg/mL (77.31 mM; Need ultrasonic).

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

References:

  1. Chen P, et al. Discovery and Characterization of GSK2801, a Selective Chemical Probe for the Bromodomains BAZ2A and BAZ2B. J Med Chem. 2016 Feb 25;59(4):1410-24.

Products are for research use only. Not for human use.

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