Description
EHMT2-IN-1 is a potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disorder or cancer.
Product information
CAS Number: 2230849-55-3
Molecular Weight: 353.42
Formula: C18H23N7O
Chemical Name: N2-(4-methoxy-3-{4-[(methylamino)methyl]-1H-pyrazol-1-yl}phenyl)-N4,6-dimethylpyrimidine-2,4-diamine
Smiles: CC1=CC(NC)=NC(NC2=CC(=C(C=C2)OC)N2C=C(CNC)C=N2)=N1
InChiKey: DJSJHTKOFPOYRZ-UHFFFAOYSA-N
InChi: InChI=1S/C18H23N7O/c1-12-7-17(20-3)24-18(22-12)23-14-5-6-16(26-4)15(8-14)25-11-13(9-19-2)10-21-25/h5-8,10-11,19H,9H2,1-4H3,(H2,20,22,23,24)
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Solubility: DMSO : 55 mg/mL (155.62 mM; Need ultrasonic).
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
How to use
In Vitro:
EHMT2-IN-1 (Compound 108) potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2.
Products are for research use only. Not for human use.
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