Perzinfotel


Catalog No. Size PriceQuantity
M18179-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

Perzinfotel (EAA-090) is a potent, selective, and competitive NMDA receptor antagonist with neuroprotective effects. Perzinfotel (EAA-090) shows high affinity (IC50=30 nM) for the glutamate site.

Product information

CAS Number: 144912-63-0

Molecular Weight: 260.18

Formula: C9H13N2O5P

Chemical Name: (2-{8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl}ethyl)phosphonic acid

Smiles: OP(O)(=O)CCN1CCCNC2=C1C(=O)C2=O

InChiKey: BDABGOLMYNHHTR-UHFFFAOYSA-N

InChi: InChI=1S/C9H13N2O5P/c12-8-6-7(9(8)13)11(3-1-2-10-6)4-5-17(14,15)16/h10H,1-5H2,(H2,14,15,16)

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Solubility: DMSO : 20.83 mg/mL (80.06 mM; Need ultrasonic). H2O : 5.88 mg/mL (22.60 mM; ultrasonic and warming and heat to 60°C).

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

How to use

In Vitro:

Perzinfotel blocks NMDA-induced currents with an IC50 of 0.48 μM and glutamate-induced neurotoxicity with an IC50 of 1.6 μM.

Products are for research use only. Not for human use.

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