Description
BIM 23056, a linear octapeptide, is a potent sst3 and sst5 somatostatin receptor antagonist with Ki values of 10.8, 5.7, respectively.
Product information
CAS Number: 150155-61-6
Molecular Weight: 1232.47
Formula: C71H81N11O9
Chemical Name: (Z,2S)-6-amino-2-[(Z)-[(2R)-2-[(Z)-[(2S)-2-[(Z)-[(2S)-2-[(Z)-[(2R)-2-amino-1-hydroxy-3-phenylpropylidene]amino]-1-hydroxy-3-phenylpropylidene]amino]-1-hydroxy-3-(4-hydroxyphenyl)propylidene]amino]-1-hydroxy-3-(1H-indol-3-yl)propylidene]amino]-N-[(1S)-1-[(Z)-[(1S)-1-[(Z)-[(1R)-1-(C-hydroxycarbonimidoyl)-2-(naphthalen-2-yl)ethyl]-C-hydroxycarbonimidoyl]-2-phenylethyl]-C-hydroxycarbonimidoyl]-2-methylpropyl]hexanimidic acid
Smiles: CC(C)[C@H](/N=C(\O)/[C@H](CCCCN)/N=C(\O)/[C@@H](CC1=CNC2=CC=CC=C21)/N=C(\O)/[C@H](CC1=CC=C(O)C=C1)/N=C(\O)/[C@H](CC1=CC=CC=C1)/N=C(\O)/[C@H](N)CC1=CC=CC=C1)/C(/O)=N/[C@@H](CC1=CC=CC=C1)/C(/O)=N/[C@H](CC1C=CC2=CC=CC=C2C=1)C(=N)O
InChiKey: VPTPBEUWKCLZGU-OOSWLFMASA-N
InChi: InChI=1S/C71H81N11O9/c1-44(2)63(71(91)81-61(39-47-22-10-5-11-23-47)67(87)77-58(64(74)84)41-49-29-32-50-24-12-13-25-51(50)36-49)82-66(86)57(28-16-17-35-72)76-70(90)62(42-52-43-75-56-27-15-14-26-54(52)56)80-69(89)60(40-48-30-33-53(83)34-31-48)79-68(88)59(38-46-20-8-4-9-21-46)78-65(85)55(73)37-45-18-6-3-7-19-45/h3-15,18-27,29-34,36,43-44,55,57-63,75,83H,16-17,28,35,37-42,72-73H2,1-2H3,(H2,74,84)(H,76,90)(H,77,87)(H,78,85)(H,79,88)(H,80,89)(H,81,91)(H,82,86)/t55-,57+,58-,59+,60+,61+,62-,63+/m1/s1
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
How to use
In Vitro:
BIM 23056 has Ki values of 142, 16.6, >1000 for sst1, sst4, sst2 , respectively.
Products are for research use only. Not for human use.
Payment & Security
Your payment information is processed securely. We do not store credit card details nor have access to your credit card information.