Linperlisib


Catalog No. Size PriceQuantity
M18300-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

Linperlisib (YY-20394) is a potent, orally bioavailable and selective inhibitor of PI3Kδ extracted from patent WO 2015055071 A1, compound 10; has an IC50 of 6.4 nM.

Product information

CAS Number: 1702816-75-8

Molecular Weight: 588.69

Formula: C28H37FN6O5S

Chemical Name: N-[5-(6-fluoro-8-{[4-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}-2-(morpholin-4-yl)quinazolin-4-yl)-2-methoxypyridin-3-yl]methanesulfonamide

Smiles: COC1=NC=C(C=C1NS(C)(=O)=O)C1N=C(N=C2C=1C=C(F)C=C2CN1CCC(CC1)C(C)(C)O)N1CCOCC1

InChiKey: NVWKNQGHVMMAJW-UHFFFAOYSA-N

InChi: InChI=1S/C28H37FN6O5S/c1-28(2,36)20-5-7-34(8-6-20)17-19-13-21(29)15-22-24(31-27(32-25(19)22)35-9-11-40-12-10-35)18-14-23(33-41(4,37)38)26(39-3)30-16-18/h13-16,20,33,36H,5-12,17H2,1-4H3

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Solubility: DMSO : 100 mg/mL (169.87 mM; Need ultrasonic).

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

How to use

In Vitro:

Linperlisib (YY-20394) is under the study for the recurrent and/or refractory follicular lymphoma.

Products are for research use only. Not for human use.

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