Description
DMP-543 (XR-543) is a KV7 channel blocker, also acts as a potent neurotransmitter release enhancer.
Product information
CAS Number: 160588-45-4
Molecular Weight: 412.43
Formula: C26H18F2N2O
Chemical Name: 10,10-bis[(2-fluoropyridin-4-yl)methyl]-9,10-dihydroanthracen-9-one
Smiles: O=C1C2=CC=CC=C2C(CC2=CC(F)=NC=C2)(CC2=CC(F)=NC=C2)C2=CC=CC=C21
InChiKey: MUJBUUDUXGDXLW-UHFFFAOYSA-N
InChi: InChI=1S/C26H18F2N2O/c27-23-13-17(9-11-29-23)15-26(16-18-10-12-30-24(28)14-18)21-7-3-1-5-19(21)25(31)20-6-2-4-8-22(20)26/h1-14H,15-16H2
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Solubility: DMSO : 100 mg/mL (242.47 mM; Need ultrasonic).
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
How to use
In Vitro:
DMP-543 enhances [3H]ACh release from rat brain slices, with an EC50 of 700 nM.
Products are for research use only. Not for human use.
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