Nav1.7-IN-2


Catalog No. Size PriceQuantity
M28131-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

Nav1.7-IN-2 is an inhibitor of voltage-gated sodium channels (Nav), in particular Nav 1.7, with IC50 of 80 nM.IC50 value: 80 nMTarget: Nav 1.7Nav1.7-IN-2 is useful for the treatment of diseases treatable by inhibition of these channels, in particular, chronic pain disorder. The more detailed information please refer to WO 2011103196 A1. Nav1.7-IN-2 is a Nav1.7 channel inhibitor extracted from patent WO/2011103196 A1, compound example J, has an IC50 of 80 nM.

Product information

CAS Number: 1332295-35-8

Molecular Weight: 407.44

Formula: C22H22FN5O2

Chemical Name: 3-({4-[3-(4-fluoro-2-methylphenoxy)azetidin-1-yl]pyrimidin-2-yl}amino)-N-methylbenzamide

Smiles: CC1=CC(F)=CC=C1OC1CN(C1)C1=CC=NC(NC2=CC(=CC=C2)C(=O)NC)=N1

InChiKey: MFAKJGXMORSMIX-UHFFFAOYSA-N

InChi: InChI=1S/C22H22FN5O2/c1-14-10-16(23)6-7-19(14)30-18-12-28(13-18)20-8-9-25-22(27-20)26-17-5-3-4-15(11-17)21(29)24-2/h3-11,18H,12-13H2,1-2H3,(H,24,29)(H,25,26,27)

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

Products are for research use only. Not for human use.

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