Description
KPLH1130 is a specific pyruvate dehydrogenase kinase (PDK) inhibitor, blocks macrophage polarization and attenuates proinflammatory responses. KPLH1130 improves glucose tolerance in HFD-fed mice.
Product information
CAS Number: 906669-07-6
Molecular Weight: 283.28
Formula: C15H13N3O3
Chemical Name: 3-(2,4-dihydroxyphenyl)-4-(4-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
Smiles: CC1C=CC(=CC=1)N1C(=O)NN=C1C1=CC=C(O)C=C1O
InChiKey: UUTBMTOBGXJTLN-UHFFFAOYSA-N
InChi: InChI=1S/C15H13N3O3/c1-9-2-4-10(5-3-9)18-14(16-17-15(18)21)12-7-6-11(19)8-13(12)20/h2-8,19-20H,1H3,(H,17,21)
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Solubility: DMSO : 135 mg/mL (476.56 mM; Need ultrasonic).
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
Products are for research use only. Not for human use.
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