Org30958


Catalog No. Size PriceQuantity
M30240-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

Org30958 is a potent aromatase inhibitor in vivo.

Product information

CAS Number: 99957-90-1

Molecular Weight: 378.59

Formula: C21H30O2S2

Chemical Name: (3aS,3bS,9aS,9bS,11aS)-9a-[(ethyldisulfanyl)methyl]-11a-methyl-1H,2H,3H,3aH,3bH,4H,5H,7H,8H,9H,9aH,9bH,10H,11H,11aH-cyclopenta[a]phenanthrene-1,7-dione

Smiles: C[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@@]43CSSCC)[C@@H]1CCC2=O

InChiKey: RCEOCOMZMSAAFR-OAGDOXAWSA-N

InChi: InChI=1S/C21H30O2S2/c1-3-24-25-13-21-11-8-15(22)12-14(21)4-5-16-17-6-7-19(23)20(17,2)10-9-18(16)21/h12,16-18H,3-11,13H2,1-2H3/t16-,17-,18-,20-,21+/m0/s1

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

How to use

In Vivo:

Besides inhibition of cornification of vaginal epithelium Org30958 (ORG 30958) decreases ovarian aromatase and plasma E2 levels in DHEAS-treated hypophysectomized rats. Plasma estradiol levels are also lowered by Org30958 in dogs which are treated with pregnant mare serum gonadotrophin in order to induce pro-estrus. Org30958 displays much less than 1/400th of the androgenic activity of testosterone propionate in immature castrated rats and appears to be devoid of estrogenic and anti-estrogenic activity in ovariectomized mature rats. A twice daily dose of 1.5 mg Org30958/kg postpones ovulation in mature female rats.

Products are for research use only. Not for human use.

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