Description
GSK3004774 is a potent, nonabsorbable agonist of CaSR, with an pEC50 of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR, respectively. GSK3004774 shows an EC50 of 50 nM for human CaSR.
Product information
CAS Number: 2138814-32-9
Molecular Weight: 528.69
Formula: C32H40N4O3
Chemical Name: 1-[3-({4-[(3R)-3-{[(1S)-1-(naphthalen-1-yl)ethyl]amino}pyrrolidin-1-yl]phenyl}formamido)propyl]piperidine-4-carboxylic acid
Smiles: C[C@H](N[C@@H]1CCN(C1)C1=CC=C(C=C1)C(=O)NCCCN1CCC(CC1)C(O)=O)C1=CC=CC2=CC=CC=C21
InChiKey: HBTVUVNVTSSIHP-WNCULLNHSA-N
InChi: InChI=1S/C32H40N4O3/c1-23(29-9-4-7-24-6-2-3-8-30(24)29)34-27-16-21-36(22-27)28-12-10-25(11-13-28)31(37)33-17-5-18-35-19-14-26(15-20-35)32(38)39/h2-4,6-13,23,26-27,34H,5,14-22H2,1H3,(H,33,37)(H,38,39)/t23-,27+/m0/s1
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
Products are for research use only. Not for human use.
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