DC_C66


Catalog No. Size PriceQuantity
M31862-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

DC_C66 is a cell-permeable, selective coactivator associated arginine methyltransferase 1 (CARM1) inhibitor with an IC50 of 1.8 μM. DC_C66 has a good selectivity for CARM1 against PRMT1 (IC50=21 μM), PRMT6 (IC50= 47μM), and PRMT5.

Product information

CAS Number: 108181-00-6

Molecular Weight: 404.48

Formula: C28H22NO2

Chemical Name: 26-(ethoxycarbonyl)-25λ⁵-azahexacyclo[12.12.0.0²,⁷.0⁸,¹³.0¹⁶,²⁵.0¹⁷,²²]hexacosa-1(26),2,4,6,8,10,12,14,16(25),17,19,21-dodecaen-25-ylium

Smiles: CCOC(=O)C1=C2C3=CC=CC=C3C3=CC=CC=C3C2=CC2C3=CC=CC=C3CC[N+]=21

InChiKey: DIVJVPWHSSAIPN-UHFFFAOYSA-N

InChi: InChI=1S/C28H22NO2/c1-2-31-28(30)27-26-23-14-8-7-12-21(23)20-11-5-6-13-22(20)24(26)17-25-19-10-4-3-9-18(19)15-16-29(25)27/h3-14,17H,2,15-16H2,1H3/q+1

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

How to use

In Vitro:

DC_C66 (6.25-100 μM; 24-72 hours) exhibits antiproliferation activity in several CARM1-associated cancer cell lines.

Products are for research use only. Not for human use.

Payment & Security

PayPal Venmo

Your payment information is processed securely. We do not store credit card details nor have access to your credit card information.

You may also like

Recently viewed