DprE1-IN-1


Catalog No. Size PriceQuantity
M33852-C Contact sales@xcessbio.com for quotation $100

Description

DprE1-IN-1 is a potent, orally active DprE1 inhibitor with favorable hepatocyte stability, low cytotoxicity and low hERG channel inhibition. DprE1-IN-1 displays potent activity aqainst both drug-susceptible and clinically isolated drug-resistant Tuberculosis strains with MICs<0.1 ug/mL. as well as good intracellular antimycobacterial activity with a 1.29 log1o CFU reduction in macrophages[1]

Product information

CAS Number: 920459-41-2

Molecular Weight: 451.52

Formula: C19H21N3O6S2

Smiles: CCOC(=O)NC(=O)C1C=CSC=1NC(=O)C1C=CC(=CC=1)S(=O)(=O)N1CCCC1

InChiKey: FFUVSZKOCCMGPX-UHFFFAOYSA-N

InChi: InChI=1S/C19H21N3O6S2/c1-2-28-19(25)21-17(24)15-9-12-29-18(15)20-16(23)13-5-7-14(8-6-13)30(26,27)22-10-3-4-11-22/h5-9,12H,2-4,10-11H2,1H3,(H,20,23)(H,21,24,25)

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Solubility: To be determined

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

Products are for research use only. Not for human use.

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