BIX 02565


Catalog No. Size PriceQuantity
M10148-2 Solid 2 mg $110
M10148-10 Solid 10 mg $330

Description

BIX 02565 is a novel RSK2 inhibitor with IC50 value of 1 nM. BIX 02565 inhibits adrenergic ɑ1A-, ɑ1B-, ɑ1D-, ɑ2A-, β2- and imidazoline I2 receptors with IC50 values ranging from 0.052 to 1.820 μM. These receptors played important roles in the regulation of vascular tone and cardiac function

Product information

CAS Number: 1311367-27-7

Molecular Weight: 458.56

Formula: C26H30N6O2

Chemical Name: (5R)-N-{1-[3-(dimethylamino)propyl]-1H-1,3-benzodiazol-2-yl}-5-methyl-1-oxo-1H,2H,3H,4H,5H-[1,4]diazepino[1,2-a]indole-8-carboxamide

Smiles: CN(C)CCCN1C(NC(=O)C2=CC3=C(C=C4C(=O)NCC[C@@H](C)N34)C=C2)=NC2=CC=CC=C12

InChiKey: ZHMXXVNQAFCXKK-QGZVFWFLSA-N

InChi: InChI=1S/C26H30N6O2/c1-17-11-12-27-25(34)23-15-18-9-10-19(16-22(18)32(17)23)24(33)29-26-28-20-7-4-5-8-21(20)31(26)14-6-13-30(2)3/h4-5,7-10,15-17H,6,11-14H2,1-3H3,(H,27,34)(H,28,29,33)/t17-/m1/s1

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥360 days if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

Products are for research use only. Not for human use.

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