Description
SB-277011, also known as SB-277011-A, is a orally active, potent and selective dopamine D(3) receptor antagonist with high oral bioavailability and CNS penetration in the rat. SB-277011-A potentiates phMRI response to acute amphetamine challenge in the rat brain. SB-277011-A attenuates ethanol consumption in ethanol preferring (P) and non-preferring (NP) rats.
Product information
CAS Number: 215803-78-4
Molecular Weight: 438.56
Formula: C28H30N4O
Chemical Name: N-{4-[2-(6-cyano-1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]cyclohexyl}quinoline-4-carboxamide
Smiles: N#CC1C=C2CCN(CC2=CC=1)CCC1CCC(CC1)NC(=O)C1=CC=NC2=CC=CC=C21
InChiKey: OLWRVVHPJFLNPW-UHFFFAOYSA-N
InChi: InChI=1S/C28H30N4O/c29-18-21-5-8-23-19-32(16-13-22(23)17-21)15-12-20-6-9-24(10-7-20)31-28(33)26-11-14-30-27-4-2-1-3-25(26)27/h1-5,8,11,14,17,20,24H,6-7,9-10,12-13,15-16,19H2,(H,31,33)
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥360 days if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
Products are for research use only. Not for human use.
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