CBP/p300 ligand 2 - CAS# 2484741-78-6


Catalog No. Size PriceQuantity
M17469-C Contact sales@xcessbio.com for quotation $100

Description

CBP/p300 ligand 2 is a ligand for target protein for PROTAC of dCBP-1. dCBP-1 is a potent and selective heterobifunctional degrader of p300/CBP.

Product information

CAS Number: 2484741-78-6

Molecular Weight: 524.61

Formula: C27H34F2N8O

Chemical Name: 3-[7-(difluoromethyl)-6-(1-methyl-1H-pyrazol-4-yl)-1, 2, 3, 4-tetrahydroquinolin-1-yl]-N-methyl-1-(piperidin-4-yl)-1H, 4H, 5H, 6H, 7H-pyrazolo[4, 3-c]pyridine-5-carboxamide

Smiles: CN1C=C(C=N1)C1=CC2CCCN(C3=NN(C4CCNCC4)C4CCN(CC=43)C(=O)NC)C=2C=C1C(F)F

InChiKey: XFGMGPKELLCGAA-UHFFFAOYSA-N

InChi: InChI=1S/C27H34F2N8O/c1-30-27(38)35-11-7-23-22(16-35)26(33-37(23)19-5-8-31-9-6-19)36-10-3-4-17-12-20(18-14-32-34(2)15-18)21(25(28)29)13-24(17)36/h12-15,19,25,31H,3-11,16H2,1-2H3,(H,30,38)

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Solubility: DMSO : 200 mg/mL (381.24 mM; Need ultrasonic).

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

How to use

In Vitro:

CBP/p300 ligand 2 (example 229) has no toxicity to LNCaP prostate cancer cells.

Products are for research use only. Not for human use.

Payment & Security

PayPal Venmo

Your payment information is processed securely. We do not store credit card details nor have access to your credit card information.

Estimate shipping

You may also like

Recently viewed