Description
RVD-Hpα TFA is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. RVD-Hpα TFA increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. RVD-Hpα TFA also high affinity CB2 positive allosteric modulator (Ki=50 nM).
Product information
Molecular Weight: 1538.67
Formula: C67H106F3N19O19
Chemical Name: (3S, 6S, 9S, 12S, 15S, 18S, 21S, 24S)-24-((1H-imidazol-4-yl)methyl)-1-((S)-1-(L-arginyl-L-valyl-L-aspartyl)pyrrolidin-2-yl)-6-(2-amino-2-oxoethyl)-12-(4-aminobutyl)-9-benzyl-21-(hydroxymethyl)-15, 18-diisobutyl-3-isopropyl-1, 4, 7, 10, 13, 16, 19, 22-octaoxo-2, 5, 8, 11, 14, 17, 20, 23-octaazapentacosan-25-oic acid--2, 2, 2-trifluoroacetic acid (1/1)
Smiles: CC(C)[C@H](NC(=O)[C@@H](N)CCCNC(N)=N)C(=O)N[C@@H](CC(O)=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC1C=CC=CC=1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC1=CNC=N1)C(O)=O.OC(=O)C(F)(F)F
InChiKey: YOAPGJLBELYWHN-WRVANEEBSA-N
InChi: InChI=1S/C65H105N19O17.C2HF3O2/c1-33(2)24-41(55(91)76-42(25-34(3)4)56(92)81-47(31-85)59(95)80-46(64(100)101)27-38-30-71-32-73-38)75-54(90)40(19-12-13-21-66)74-57(93)43(26-37-16-10-9-11-17-37)77-58(94)44(28-49(68)86)78-61(97)52(36(7)8)83-60(96)48-20-15-23-84(48)63(99)45(29-50(87)88)79-62(98)51(35(5)6)82-53(89)39(67)18-14-22-72-65(69)70;3-2(4,5)1(6)7/h9-11,16-17,30,32-36,39-48,51-52,85H,12-15,18-29,31,66-67H2,1-8H3,(H2,68,86)(H,71,73)(H,74,93)(H,75,90)(H,76,91)(H,77,94)(H,78,97)(H,79,98)(H,80,95)(H,81,92)(H,82,89)(H,83,96)(H,87,88)(H,100,101)(H4,69,70,72);(H,6,7)/t39-,40-,41-,42-,43-,44-,45-,46-,47-,48-,51-,52-;/m0./s1
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
Products are for research use only. Not for human use.
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