Description
GS-626510 is a potent, and orally active BET family bromodomains inhibitor, with Kd values of 0.59-3.2 nM for BRD2/3/4, with IC50 values of 83 nM and 78 nM foe BD1 and BD2, respectively.
Product information
CAS Number: 1637770-13-8
Molecular Weight: 394.47
Formula: C25H22N4O
Chemical Name: 5-[2-cyclopropyl-5-(3,5-dimethyl-1,2-oxazol-4-yl)-1H-1,3-benzodiazol-7-yl]-6-methylquinoline
Smiles: CC1=CC=C2N=CC=CC2=C1C1C=C(C=C2N=C(NC=12)C1CC1)C1C(C)=NOC=1C
InChiKey: KHQQNXFBTALTQF-UHFFFAOYSA-N
InChi: InChI=1S/C25H22N4O/c1-13-6-9-20-18(5-4-10-26-20)22(13)19-11-17(23-14(2)29-30-15(23)3)12-21-24(19)28-25(27-21)16-7-8-16/h4-6,9-12,16H,7-8H2,1-3H3,(H,27,28)
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Solubility: DMSO : 25 mg/mL (63.38 mM; ultrasonic and warming and adjust pH to 4 with HCl and heat to 80°C).
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
Products are for research use only. Not for human use.
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