GS-626510


Catalog No. Size PriceQuantity
M17883-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

GS-626510 is a potent, and orally active BET family bromodomains inhibitor, with Kd values of 0.59-3.2 nM for BRD2/3/4, with IC50 values of 83 nM and 78 nM foe BD1 and BD2, respectively.

Product information

CAS Number: 1637770-13-8

Molecular Weight: 394.47

Formula: C25H22N4O

Chemical Name: 5-[2-cyclopropyl-5-(3,5-dimethyl-1,2-oxazol-4-yl)-1H-1,3-benzodiazol-7-yl]-6-methylquinoline

Smiles: CC1=CC=C2N=CC=CC2=C1C1C=C(C=C2N=C(NC=12)C1CC1)C1C(C)=NOC=1C

InChiKey: KHQQNXFBTALTQF-UHFFFAOYSA-N

InChi: InChI=1S/C25H22N4O/c1-13-6-9-20-18(5-4-10-26-20)22(13)19-11-17(23-14(2)29-30-15(23)3)12-21-24(19)28-25(27-21)16-7-8-16/h4-6,9-12,16H,7-8H2,1-3H3,(H,27,28)

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Solubility: DMSO : 25 mg/mL (63.38 mM; ultrasonic and warming and adjust pH to 4 with HCl and heat to 80°C).

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

Products are for research use only. Not for human use.

Payment & Security

PayPal Venmo

Your payment information is processed securely. We do not store credit card details nor have access to your credit card information.

You may also like

Recently viewed