Description
EHMT2-IN-2 is a potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disease or cancer.
Product information
CAS Number: 2230850-47-0
Molecular Weight: 374.44
Formula: C21H22N6O
Chemical Name: N2-(4-methoxy-3-{3-methyl-1H-pyrrolo[2,3-c]pyridin-2-yl}phenyl)-N4,6-dimethylpyrimidine-2,4-diamine
Smiles: CNC1C=C(C)N=C(NC2C=C(C3NC4C=NC=CC=4C=3C)C(=CC=2)OC)N=1
InChiKey: AZRYONWATLLNFX-UHFFFAOYSA-N
InChi: InChI=1S/C21H22N6O/c1-12-9-19(22-3)27-21(24-12)25-14-5-6-18(28-4)16(10-14)20-13(2)15-7-8-23-11-17(15)26-20/h5-11,26H,1-4H3,(H2,22,24,25,27)
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
How to use
In Vitro:
EHMT2-IN-2 (Compound 200) is a potent EHMT inhibitor, with IC50s of all < 100 nM for EEHMT1 peptide, EHMT2 peptide and cellular EHMT2.
Products are for research use only. Not for human use.
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