Halopemide


Catalog No. Size PriceQuantity
M18751-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

Halopemide is a potent phospholipase D (PLD) inhibitor, with IC50s of 220 and 310 nM for human PLD1 and PLD2, respectively. Halopemid is a dopamine receptors antagonist, and acts a psychotropic agent.

Product information

CAS Number: 59831-65-1

Molecular Weight: 416.88

Formula: C21H22ClFN4O2

Chemical Name: N-{2-[4-(5-chloro-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]ethyl}-4-fluorobenzamide

Smiles: O=C1NC2C=C(Cl)C=CC=2N1C1CCN(CCNC(=O)C2C=CC(F)=CC=2)CC1

InChiKey: NBHPRWLFLUBAIE-UHFFFAOYSA-N

InChi: InChI=1S/C21H22ClFN4O2/c22-15-3-6-19-18(13-15)25-21(29)27(19)17-7-10-26(11-8-17)12-9-24-20(28)14-1-4-16(23)5-2-14/h1-6,13,17H,7-12H2,(H,24,28)(H,25,29)

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

How to use

In Vitro:

Halopemide (1-2 μM; 21 day) affects calcification in transdifferentiated MOVAS cells.

In Vivo:

Halopemide (10 mg/kg; p.o.) induces dyskinesias in the majority of monkeys tested.

Products are for research use only. Not for human use.

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