Rocastine


Catalog No. Size PriceQuantity
M19497-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

Rocastine is a selective, nonsedating H1 antagonist, acting as an antihistamine.

Product information

CAS Number: 91833-49-7

Molecular Weight: 265.37

Formula: C13H19N3OS

Chemical Name: 2-[2-(dimethylamino)ethyl]-4-methyl-2H,3H,4H,5H-pyrido[3,2-f][1,4]oxazepine-5-thione

Smiles: CN(C)CCC1CN(C)C(=S)C2=CC=CN=C2O1

InChiKey: DPPDPATYPQFYDL-UHFFFAOYSA-N

InChi: InChI=1S/C13H19N3OS/c1-15(2)8-6-10-9-16(3)13(18)11-5-4-7-14-12(11)17-10/h4-5,7,10H,6,8-9H2,1-3H3

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

How to use

In Vivo:

Rocastine is effective with a 15 min pretreatment time (PD50 = 0.13 mg/kg) as it is with a 1 hr pretreatment time (PD50 = 0.12 mg/kg). Rocastine protects guinea pigs from collapse induced by aerosolized antigen; rocastine is approximately 36x more potent than diphenhydramine and as potent as oxatomide and terfenadine. Rocastine does not alter the EEG of cats at doses in vast excess (150x) of its antihistaminic dose nor does it potentiate yohimbine toxicity in mice.

Products are for research use only. Not for human use.

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