GSK9027


Catalog No. Size PriceQuantity
M21488-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

GSK9027, as a non-steroidal glucocorticoid receptor (GR) agonist, behaves as a partial agonist on the 2×glucocorticoid response element (GRE) reporter system, and achieves intrinsic activities relative to dexamethasone.

Product information

CAS Number: 1229096-88-1

Molecular Weight: 525.52

Formula: C27H19F4N3O2S

Chemical Name: N-{4-[1-(4-fluorophenyl)-1H-indazol-5-yl]-3-(trifluoromethyl)phenyl}-1-phenylmethanesulfonamide

Smiles: O=S(=O)(CC1C=CC=CC=1)NC1=CC(=C(C=C1)C1C=C2C=NN(C3=CC=C(F)C=C3)C2=CC=1)C(F)(F)F

InChiKey: DXBJGDVBQPEMOB-UHFFFAOYSA-N

InChi: InChI=1S/C27H19F4N3O2S/c28-21-7-10-23(11-8-21)34-26-13-6-19(14-20(26)16-32-34)24-12-9-22(15-25(24)27(29,30)31)33-37(35,36)17-18-4-2-1-3-5-18/h1-16,33H,17H2

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

How to use

In Vitro:

GSK9027 demonstrates reduced 2×GRE reporter activation and is partial agonists.

Products are for research use only. Not for human use.

Payment & Security

PayPal Venmo

Your payment information is processed securely. We do not store credit card details nor have access to your credit card information.

You may also like

Recently viewed