GSK805


Catalog No. Size PriceQuantity
M21652-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

GSK805 is a potent, orally bioavailable, and CNS penetrant RORγt inhibitor with pIC50 of 8.4 and >8.2 for RORγ FRET assay and Th17 assay.

Product information

CAS Number: 1426802-50-7

Molecular Weight: 532.36

Formula: C23H18Cl2F3NO4S

Chemical Name: N-[2,6-dichloro-2'-(trifluoromethoxy)-[1,1'-biphenyl]-4-yl]-2-[4-(ethanesulfonyl)phenyl]acetamide

Smiles: CCS(=O)(=O)C1C=CC(CC(=O)NC2C=C(Cl)C(=C(Cl)C=2)C2C=CC=CC=2OC(F)(F)F)=CC=1

InChiKey: CEICQMBWAQAIQX-UHFFFAOYSA-N

InChi: InChI=1S/C23H18Cl2F3NO4S/c1-2-34(31,32)16-9-7-14(8-10-16)11-21(30)29-15-12-18(24)22(19(25)13-15)17-5-3-4-6-20(17)33-23(26,27)28/h3-10,12-13H,2,11H2,1H3,(H,29,30)

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Solubility: DMSO : ≥ 100 mg/mL (187.84 mM).

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

Products are for research use only. Not for human use.

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