Description
Pipequaline (PK 8165) is a partial benzodiazepine receptor agonist with anxiolytic activity.
Product information
CAS Number: 77472-98-1
Molecular Weight: 316.44
Formula: C22H24N2
Chemical Name: 2-phenyl-4-[2-(piperidin-4-yl)ethyl]quinoline
Smiles: C(CC1CCNCC1)C1=CC(=NC2=CC=CC=C12)C1C=CC=CC=1
InChiKey: AMEWZCMTSIONOX-UHFFFAOYSA-N
InChi: InChI=1S/C22H24N2/c1-2-6-18(7-3-1)22-16-19(11-10-17-12-14-23-15-13-17)20-8-4-5-9-21(20)24-22/h1-9,16-17,23H,10-15H2
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Solubility: DMSO : ≥ 32 mg/mL (101.13 mM).
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
How to use
In Vivo:
Intravenously administered pipequaline exerts a partial suppression of activations by kainate, glutamate and acetylcholine. Microiontophoretic applications of pipequaline reduces the neuronal activation by kainate. Pipequaline produces dose-related decreases in motor activity. Pipequaline produces significant dose-related decreases in the number of head-dips made.
Products are for research use only. Not for human use.
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