Asperphenamate


Catalog No. Size PriceQuantity
M23883-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

Asperphenamate, a fungal metabolite of Aspergillus flatiipes with anti-cancer effect, exhibits IC50 values of 92.3 μM, 96.5 μM and 97.9 μM in T47D, MDA-MB-231 and HL-60 cells, respectively.

Product information

CAS Number: 63631-36-7

Molecular Weight: 506.59

Formula: C32H30N2O4

Chemical Name: (2S)-3-phenyl-2-(phenylformamido)propyl (2S)-3-phenyl-2-(phenylformamido)propanoate

Smiles: O=C(N[C@H](COC(=O)[C@H](CC1C=CC=CC=1)NC(=O)C1C=CC=CC=1)CC1C=CC=CC=1)C1C=CC=CC=1

InChiKey: CVULDJMCSSACEO-VMPREFPWSA-N

InChi: InChI=1S/C32H30N2O4/c35-30(26-17-9-3-10-18-26)33-28(21-24-13-5-1-6-14-24)23-38-32(37)29(22-25-15-7-2-8-16-25)34-31(36)27-19-11-4-12-20-27/h1-20,28-29H,21-23H2,(H,33,35)(H,34,36)/t28-,29-/m0/s1

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Solubility: DMSO : 100 mg/mL (197.40 mM; Need ultrasonic).

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

How to use

In Vitro:

Asperphenamate can inhibit cancer cell proliferation by fully inducing autophagy. asperphenamate showed inhibition effects against cathepsin L. At the same time, it also displayed weak inhibitory ability against cathepsin S.

Products are for research use only. Not for human use.

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