Description
PF-06795071 is a potent and selective covalent MAGL inhibitor with an IC50 of 3 nM.
Product information
CAS Number: 2075629-81-9
Molecular Weight: 399.34
Formula: C18H17F4N3O3
Chemical Name: (2R)-1,1,1-trifluoro-3-hydroxypropan-2-yl (1R,5S)-6-[1-(4-fluorophenyl)-1H-pyrazol-3-yl]-3-azabicyclo[3.1.0]hexane-3-carboxylate
Smiles: OC[C@@H](OC(=O)N1C[C@@H]2C([C@@H]2C1)C1C=CN(N=1)C1=CC=C(F)C=C1)C(F)(F)F
InChiKey: MEDCQBUTCWNKGW-XFDYKOMQSA-N
InChi: InChI=1S/C18H17F4N3O3/c19-10-1-3-11(4-2-10)25-6-5-14(23-25)16-12-7-24(8-13(12)16)17(27)28-15(9-26)18(20,21)22/h1-6,12-13,15-16,26H,7-9H2/t12-,13+,15-,16?/m1/s1
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
How to use
In Vitro:
PF-06795071 shows excellent selectivity against FAAH with an IC50 of 3.1 μM.
Products are for research use only. Not for human use.
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