AZ-Dyrk1B-33


Catalog No. Size PriceQuantity
M27181-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

AZ-Dyrk1B-33 is a potent and selective Dyrk1B kinase inhibitor, with an IC50 of 7 nM.

Product information

CAS Number: 1679330-37-0

Molecular Weight: 300.36

Formula: C19H16N4

Chemical Name: 4-{1-benzyl-1H-pyrrolo[2,3-c]pyridin-3-yl}-2-methylpyrimidine

Smiles: CC1=NC(=CC=N1)C1=CN(CC2C=CC=CC=2)C2=CN=CC=C21

InChiKey: CZCUSHJQJWKYTD-UHFFFAOYSA-N

InChi: InChI=1S/C19H16N4/c1-14-21-10-8-18(22-14)17-13-23(12-15-5-3-2-4-6-15)19-11-20-9-7-16(17)19/h2-11,13H,12H2,1H3

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Solubility: DMSO : 125 mg/mL (416.17 mM; Need ultrasonic).

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

How to use

In Vitro:

AZ-Dyrk1B-33 shows inhibition of phosphorylation of Dyrk pS421 in cells with an IC50 of 0.192 μM. AZ-Dyrk1B-33 shows no effect in sensitization.

Products are for research use only. Not for human use.

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