Description
PGAM1-IN-2 is a phosphoglycerate mutase 1 (PGAM1) inhibitor with an IC50 of 2.1 μM.
Product information
CAS Number: 2438637-66-0
Molecular Weight: 488.47
Formula: C25H16N2O7S
Chemical Name: N-(1-hydroxy-7-nitro-9-oxo-9H-xanthen-3-yl)-[1,1'-biphenyl]-4-sulfonamide
Smiles: [O-][N+](=O)C1=CC2=C(C=C1)OC1=CC(=CC(O)=C1C2=O)NS(=O)(=O)C1C=CC(=CC=1)C1C=CC=CC=1
InChiKey: BRBFEAYMCMDULD-UHFFFAOYSA-N
InChi: InChI=1S/C25H16N2O7S/c28-21-12-17(13-23-24(21)25(29)20-14-18(27(30)31)8-11-22(20)34-23)26-35(32,33)19-9-6-16(7-10-19)15-4-2-1-3-5-15/h1-14,26,28H
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Solubility: DMSO : 62.5 mg/mL (127.95 mM; Need ultrasonic).
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
How to use
In Vitro:
PGAM1-IN-2 (Compound 15h) inhibits H1299 proliferation with an IC50 of 33.8±6.1 μM.
Products are for research use only. Not for human use.
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