GI-530159


Catalog No. Size PriceQuantity
M28617-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

GI-530159 is a selective, mechanosensitive opener of TREK1 (K2P2.1) and TREK2 (K2P10.1) channels, with an EC50 of 0.76 μM for TREK1. GI-530159 displays selectivity for TREK1/2 over TRAAK, TASK3 and other potassium channels. GI-530159 reduces rat dorsal root ganglion neuron excitability.

Product information

CAS Number: 69563-88-8

Molecular Weight: 518.45

Formula: C27H20F6N2O2

Chemical Name: 4-(4-{2-[4-(4-aminophenoxy)phenyl]-1,1,1,3,3,3-hexafluoropropan-2-yl}phenoxy)aniline

Smiles: NC1C=CC(=CC=1)OC1C=CC(=CC=1)C(C1C=CC(=CC=1)OC1C=CC(N)=CC=1)(C(F)(F)F)C(F)(F)F

InChiKey: HHLMWQDRYZAENA-UHFFFAOYSA-N

InChi: InChI=1S/C27H20F6N2O2/c28-26(29,30)25(27(31,32)33,17-1-9-21(10-2-17)36-23-13-5-19(34)6-14-23)18-3-11-22(12-4-18)37-24-15-7-20(35)8-16-24/h1-16H,34-35H2

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Solubility: DMSO : 250 mg/mL (482.21 mM; Need ultrasonic).

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

Products are for research use only. Not for human use.

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