Description
PIK-108 is a non-ATP competitive, allosteric p110β/p110δ selective inhibitor.
Product information
CAS Number: 901398-68-3
Molecular Weight: 364.44
Formula: C22H24N2O3
Chemical Name: 6-methyl-2-(morpholin-4-yl)-8-[1-(phenylamino)ethyl]-4H-chromen-4-one
Smiles: CC1C=C2C(OC(=CC2=O)N2CCOCC2)=C(C=1)C(C)NC1C=CC=CC=1
InChiKey: VRCXIJAYLCUSHC-UHFFFAOYSA-N
InChi: InChI=1S/C22H24N2O3/c1-15-12-18(16(2)23-17-6-4-3-5-7-17)22-19(13-15)20(25)14-21(27-22)24-8-10-26-11-9-24/h3-7,12-14,16,23H,8-11H2,1-2H3
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Solubility: DMSO : 50 mg/mL (137.20 mM; Need ultrasonic).
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
How to use
In Vitro:
PIK-108 (0.1-10 μM; 1 hour) blocks phosphorylation of PKB/Akt.
Products are for research use only. Not for human use.
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