Description
CAY10698 (compound 1) is a potent and selective inhibitor of 12-Lipoxygenase (12-LOX) with an IC50 of 5.1 μM. CAY10698 is inactive against 5-LOX, 15-LOX-1, 15-LOX-2 and COX-1/2.
Product information
CAS Number: 684236-01-9
Molecular Weight: 391.46
Formula: C17H17N3O4S2
Chemical Name: 4-{[(2-hydroxy-3-methoxyphenyl)methyl]amino}-N-(1,3-thiazol-2-yl)benzene-1-sulfonamide
Smiles: COC1=CC=CC(CNC2=CC=C(C=C2)S(=O)(=O)NC2=NC=CS2)=C1O
InChiKey: CENSVXZQMJBVHY-UHFFFAOYSA-N
InChi: InChI=1S/C17H17N3O4S2/c1-24-15-4-2-3-12(16(15)21)11-19-13-5-7-14(8-6-13)26(22,23)20-17-18-9-10-25-17/h2-10,19,21H,11H2,1H3,(H,18,20)
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Solubility: DMSO : 125 mg/mL (319.32 mM; Need ultrasonic).
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
Products are for research use only. Not for human use.
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