GSK3004774


Catalog No. Size PriceQuantity
M30832-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

GSK3004774 is a potent, nonabsorbable agonist of CaSR, with an pEC50 of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR, respectively. GSK3004774 shows an EC50 of 50 nM for human CaSR.

Product information

CAS Number: 2138814-32-9

Molecular Weight: 528.69

Formula: C32H40N4O3

Chemical Name: 1-[3-({4-[(3R)-3-{[(1S)-1-(naphthalen-1-yl)ethyl]amino}pyrrolidin-1-yl]phenyl}formamido)propyl]piperidine-4-carboxylic acid

Smiles: C[C@H](N[C@@H]1CCN(C1)C1=CC=C(C=C1)C(=O)NCCCN1CCC(CC1)C(O)=O)C1=CC=CC2=CC=CC=C21

InChiKey: HBTVUVNVTSSIHP-WNCULLNHSA-N

InChi: InChI=1S/C32H40N4O3/c1-23(29-9-4-7-24-6-2-3-8-30(24)29)34-27-16-21-36(22-27)28-12-10-25(11-13-28)31(37)33-17-5-18-35-19-14-26(15-20-35)32(38)39/h2-4,6-13,23,26-27,34H,5,14-22H2,1H3,(H,33,37)(H,38,39)/t23-,27+/m0/s1

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

Products are for research use only. Not for human use.

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