Description
CCRP2, also known as TLX agonist 1 and SUN23314, is an orphan nuclear receptor tailless (TLX, NR2E1) modulator (EC50=1μM; Kd= 650 nM). TLX agonist 1 potentiates TLX transcriptional repressive activity. CCRP2 was reported in PLoS One . 2014 Jun 17;9(6):e99440.
Product information
CAS Number: 958323-31-4
Molecular Weight: 374.48
Formula: C23H26N4O
Synonym:
SUN-23314
CCRP-2
TLX agonist 1
SUN23314
SUN 23314
CCRP2
CCRP 2
Chemical Name: (4-benzhydrylpiperazin-1-yl)(1,5-dimethyl-1H-pyrazol-3-yl)methanone
Smiles: CN1N=C(C=C1C)C(=O)N1CCN(CC1)C(C1C=CC=CC=1)C1C=CC=CC=1
InChiKey: SSGJAUSSGPIZEE-UHFFFAOYSA-N
InChi: InChI=1S/C23H26N4O/c1-18-17-21(24-25(18)2)23(28)27-15-13-26(14-16-27)22(19-9-5-3-6-10-19)20-11-7-4-8-12-20/h3-12,17,22H,13-16H2,1-2H3
Technical Data
Appearance: Solid Power.
Purity: ≥98% (or refer to the Certificate of Analysis)
Solubility: Soluble in DMSO
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥360 days if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined.
HS Tariff Code: 382200
References:
- Benod C, Villagomez R, Filgueira CS, et al. The human orphan nuclear receptor tailless (TLX, NR2E1) is druggable. PLoS One. 2014;9(6):e99440. Published 2014 Jun 17. doi:10.1371/journal.pone.0099440
Products are for research use only. Not for human use.
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