CCRP2


Catalog No. size PriceQuantity
M7108-2 2mg solid $142
M7108-10 10mg solid $570

Description

Cas:958323-31-4 (free base)

Product Information

CCRP2, also known as TLX agonist 1 and SUN23314, is an orphan nuclear receptor tailless (TLX, NR2E1) modulator (EC50=1μM; Kd= 650 nM). TLX agonist 1 potentiates TLX transcriptional repressive activity. CCRP2 was reported in PLoS One . 2014 Jun 17;9(6):e99440.

 

Chemical Formula: C23H26N4O

 

Exact Mass: 374.2107

 

Molecular Weight: 374.488

 

Elemental Analysis: C, 73.77; H, 7.00; N, 14.96; O, 4.27

 

Synonym:

 

TLX agonist 1

SUN23314

SUN-23314

SUN 23314

CCRP2

CCRP-2

CCRP 2

 

Chemical Name: (4-benzhydrylpiperazin-1-yl)(1,5-dimethyl-1H-pyrazol-3-yl)methanone

 

InChi Key:

SSGJAUSSGPIZEE-UHFFFAOYSA-N

 

InChi Code: InChI=1S/C23H26N4O/c1-18-17-21(24-25(18)2)23(28)27-15-13-26(14-16-27)22(19-9-5-3-6-10-19)20-11-7-4-8-12-20/h3-12,17,22H,13-16H2,1-2H3

 

Smiles Code:

O=C(C1=NN(C)C(C)=C1)N2CCN(C(C3=CC=CC=C3)C4=CC=CC=C4)CC2

 

 

Technical Data:

 

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >3 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

 

 

References

 

  1. Benod C, Villagomez R, Filgueira CS, et al. The human orphan nuclear receptor tailless (TLX, NR2E1) is druggable. PLoS One. 2014;9(6):e99440. Published 2014 Jun 17. doi:10.1371/journal.pone.0099440

 

Products are for research use only. Not for human use.

 

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