Description
VU0119498 is a pan Gq muscarinic acetylcholine receptor (mAChR) M1, M3, M5 positive allosteric modulator (PAM) with EC50 of 6.1 μM, 6.4 μM, 4.1 μM, respectively.
Product information
CAS Number: 79183-37-2
Molecular Weight: 316.15
Formula: C15H10BrNO2
Synonym:
VU 0119498
VU-0119498
Chemical Name: 1-[(4-bromophenyl)methyl]indole-2,3-dione
Smiles: O=C1C2=CC=CC=C2N(CC2C=CC(Br)=CC=2)C1=O
InChiKey: DELLOEULSHGYCG-UHFFFAOYSA-N
InChi: InChI=1S/C15H10BrNO2/c16-11-7-5-10(6-8-11)9-17-13-4-2-1-3-12(13)14(18)15(17)19/h1-8H,9H2
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Solubility: DMSO 50 mg/mL (158.15 mM)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
References:
- Thomas M Bridges, et al. Bioorg Med Chem Lett. 2010 Mar 15;
Products are for research use only. Not for human use.
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