Description
GSK5182, 4-hydroxytamoxifen analog, is a specific inverse agonist of estrogen-related receptor γ (ERRγ) that inhibits pro-inflammatory cytokine-induced catabolic factors.
Product information
CAS Number: 877387-37-6
Molecular Weight: 417.54
Formula: C27H31NO3
Synonym:
GSK 5182
GSK-5182
Related CAS Number:
1936468-29-9 (GSK5182 (HCl))
Chemical Name: 4-[(Z)-1-[4-(2-dimethylaminoethoxy)phenyl]-5-hydroxy-2-phenylpent-1-enyl]phenol
Smiles: CN(C)CCOC1C=CC(=CC=1)/C(/C1=CC=C(O)C=C1)=C(/CCCO)\C1C=CC=CC=1
InChiKey: ZVSFNBNLNLXEFQ-RQZHXJHFSA-N
InChi: InChI=1S/C27H31NO3/c1-28(2)18-20-31-25-16-12-23(13-17-25)27(22-10-14-24(30)15-11-22)26(9-6-19-29)21-7-4-3-5-8-21/h3-5,7-8,10-17,29-30H,6,9,18-20H2,1-2H3/b27-26-
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Solubility: DMSO: 84 mg/mL(201.17 mM).
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
References:
- Yunhui Min, et al. Pharmaceuticals (Basel). 2020 Nov 27;13(12):429.
Products are for research use only. Not for human use.
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