Enpp-1-IN-1

Enpp-1-IN-1 (UUN28589, MV 658) is an inhibitor of Ectonucleotide pyrophosphatase-phosphodiesterase 1 (enpp-1).

Product information

CAS Number: 2289728-58-9

Molecular Weight: 343.40

Formula: C17H17N3O3S

Synonym:

UUN-28589

MV-658

Chemical Name: N-{[4-(7-methoxyquinolin-4-yl)phenyl]methyl}aminosulfonamide

Smiles: COC1=CC2=NC=CC(=C2C=C1)C1C=CC(CNS(N)(=O)=O)=CC=1

InChiKey: UEJMNZDIQDULLP-UHFFFAOYSA-N

InChi: InChI=1S/C17H17N3O3S/c1-23-14-6-7-16-15(8-9-19-17(16)10-14)13-4-2-12(3-5-13)11-20-24(18,21)22/h2-10,20H,11H2,1H3,(H2,18,21,22)

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Solubility: DMSO: 250 mg/mL (728.01 mM)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 ^oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 ^oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

References:

1. Preparation quinolinyl and quinazolinyl benzenesulfamides and analogs as ectonucleotide pyrophosphatase-​phosphodiesterase 1 (ENPP-​1) inhibitors as antitumor antiviral By Gallatin, William Michael; Odingo, Joshua; Dietsch, Gregory N.; Florio, Vincent; Venkateshappa, Chandregowda; Duraiswamy, Athisayamani Jeyaraj From PCT Int. Appl. (2019), WO 2019046778 A1 20190307.

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